SCHEMBL4586191

SCHEMBL4586191

O=C1N=C(Nc2cc(NC(=O)C3CCC3)ccc2Cl)SC1=Cc1ccc2ncc(C(=O)OC(=O)C(F)(F)F)c(N3CCOCC3)c2c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
TSHR P16473 1/20 0.37
GBA1 P04062 4/20 0.36
GLA P06280 1/20 0.36
EGFR P00533 3/20 0.36
MELK Q14680 7/20 0.35
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HSD17B10 Q99714 1/20 0.34
GAA P10253 1/20 0.34
ESR1 P03372 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CHRM4 P08173 1/20 0.33
SHMT2 P34897 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4586182 0.91 GBA1 (0.39) ALDH1A1HPGDTSHRGBA1GLA
Trifluoroacetic Acid SCHEMBL4586199 0.91 GBA1 (0.39) ALDH1A1HPGDTSHRGBA1GLA
Trifluoroacetic Acid SCHEMBL2988928 0.90 GAA (0.43) GBA1GLAMAPTHSD17B10GAA
Trifluoroacetic Acid SCHEMBL5049855 0.90 GAA (0.43) GBA1GLAMAPTHSD17B10GAA
SCHEMBL4585828 0.89 GAA (0.35) ALDH1A1MELKMAPTHSD17B10GAA
SCHEMBL4585472 0.83 MEN1 (0.35) EGFRESR1MEN1KMT2A
SCHEMBL4585717 0.83 MEN1 (0.38) ALDH1A1MELKKDM4EMEN1KMT2A
SCHEMBL2993692 0.83 ALDH1A1 (0.46) ALDH1A1HPGDTSHRGBA1GLA
SCHEMBL2993695 0.83 ALDH1A1 (0.46) ALDH1A1HPGDTSHRGBA1GLA
Trifluoroacetic Acid SCHEMBL2988931 0.82 GBA1 (0.39) ALDH1A1HPGDTSHRGBA1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879563-A4 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2008-07-16 EP disclosed
EP-1879563-A2 NOVEL CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-01-23 EP disclosed
WO-2006132739-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-12-14 WO disclosed