SCHEMBL4585828

SCHEMBL4585828

CC(C)C(=O)Nc1ccc(Cl)c(NC2=NC(=O)C(=Cc3ccc4ncc(C(=O)OC(=O)C(F)(F)F)c(N5CCOCC5)c4c3)S2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 6/20 0.35
MAPT P10636 6/20 0.35
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
SMN1; SMN2 Q16637 3/20 0.33
ALDH1A1 P00352 1/20 0.33
PKM P14618 1/20 0.33
BRAF P15056 1/20 0.33
LMNA P02545 2/20 0.33
MC4R P32245 2/20 0.33
HTT P42858 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
PTK2B Q14289 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MAPK1 P28482 2/20 0.32
CLK1 P49759 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
TP53 P04637 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4585717 0.93 MEN1 (0.38) MEN1KMT2AALDH1A1BRAFLMNA
Trifluoroacetic Acid SCHEMBL4585836 0.91 MEN1 (0.37) GAAMAPTMEN1KMT2ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL4585816 0.91 MEN1 (0.37) GAAMAPTMEN1KMT2ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL2990672 0.91 MAPT (0.43) GAAMAPTMEN1KMT2ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL5048576 0.91 MAPT (0.43) GAAMAPTMEN1KMT2ASMN1; SMN2
SCHEMBL4586191 0.89 ALDH1A1 (0.37) GAAMAPTMEN1KMT2AALDH1A1
Trifluoroacetic Acid SCHEMBL5048553 0.84 MEN1 (0.47) GAAMAPTMEN1KMT2AALDH1A1
Trifluoroacetic Acid SCHEMBL2988374 0.84 MEN1 (0.47) GAAMAPTMEN1KMT2AALDH1A1
Trifluoroacetic Acid SCHEMBL4585709 0.84 ENPP2 (0.39) MAPTMEN1KMT2AALDH1A1BRAF
Trifluoroacetic Acid SCHEMBL4585722 0.84 ENPP2 (0.39) MAPTMEN1KMT2AALDH1A1BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879563-A4 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2008-07-16 EP disclosed
EP-1879563-A2 NOVEL CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-01-23 EP disclosed
WO-2006132739-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-12-14 WO disclosed