SCHEMBL4586942

SCHEMBL4586942

Cc1ncnc(C)c1C(=O)NC(C)CCN1CCC(N(Cc2cc(Cl)ccc2F)c2ccc(C(=O)O)cc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 15/20 0.42
KCNH2 Q12809 2/20 0.36
PGR P06401 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
PLD2 O14939 1/20 0.35
PLD1 Q13393 1/20 0.35
SCN1A P35498 1/20 0.35
SCN8A Q9UQD0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586088 0.88 CCR5 (0.42) CCR5KCNH2PGRCYP2D6CYP2C9
SCHEMBL4586676 0.87 CCR5 (0.40) CCR5KCNH2PGRCYP2D6CYP2C9
SCHEMBL4586245 0.86 CCR5 (0.42) CCR5
SCHEMBL4244786 0.84 CCR5 (0.60) CCR5KCNH2
SCHEMBL4586504 0.81 CCR5 (0.56) CCR5
SCHEMBL4586174 0.81 CCR5 (0.43) CCR5
SCHEMBL4586981 0.81 CCR5 (0.49) CCR5KCNH2
SCHEMBL4585509 0.80 CCR5 (0.38) CCR5PGRCYP2D6CYP2C9
SCHEMBL4585280 0.79 CCR5 (0.48) CCR5PGR
SCHEMBL4587024 0.79 CCR5 (0.44) CCR5PGRCYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed