SCHEMBL4586504

SCHEMBL4586504

Cc1ncnc(C)c1C(=O)NC(C)CCN1CCC(N(Cc2ccccc2)c2ccc(Oc3ccc(C(=O)O)cc3)cc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 12/20 0.56
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44
CACNA1B Q00975 2/20 0.44
LTA4H P09960 4/20 0.43
OPRM1 P35372 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4587594 0.91 CCR5 (0.48) CCR5DRD2DRD3CACNA1B
SCHEMBL4586072 0.91 CCR5 (0.57) CCR5DRD2DRD3CACNA1BLTA4H
SCHEMBL4586981 0.86 CCR5 (0.49) CCR5DRD2DRD3
SCHEMBL4586245 0.84 CCR5 (0.42) CCR5
SCHEMBL4585297 0.84 CCR5 (0.48) CCR5DRD2DRD3CACNA1BOPRM1
SCHEMBL4241170 0.84 CCR5 (0.79) CCR5
SCHEMBL4587438 0.81 CCR5 (0.50) CCR5CACNA1B
SCHEMBL4586942 0.81 CCR5 (0.42) CCR5
SCHEMBL4586351 0.81 CCR5 (0.51) CCR5CACNA1B
SCHEMBL4586422 0.81 CCR5 (0.47) CCR5DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP claimed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP claimed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO claimed
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed