SCHEMBL4587438

SCHEMBL4587438

Cc1ncnc(C)c1C(=O)NC(C)CCN1CCC(N(Cc2cccc(C#N)c2)c2ccc(OCC(=O)O)cc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 18/20 0.50
KCNH2 Q12809 1/20 0.41
CACNA1B Q00975 1/20 0.40
DCUN1D1 Q96GG9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586351 0.92 CCR5 (0.51) CCR5KCNH2CACNA1B
SCHEMBL4586809 0.92 CCR5 (0.50) CCR5KCNH2CACNA1BDCUN1D1
SCHEMBL4587594 0.91 CCR5 (0.48) CCR5KCNH2CACNA1BDCUN1D1
SCHEMBL4585956 0.91 CCR5 (0.49) CCR5KCNH2CACNA1B
SCHEMBL4586981 0.91 CCR5 (0.49) CCR5KCNH2DCUN1D1
SCHEMBL4586733 0.91 CCR5 (0.49) CCR5KCNH2CACNA1B
SCHEMBL4586174 0.89 CCR5 (0.43) CCR5
SCHEMBL4588198 0.87 CCR5 (0.61) CCR5KCNH2CACNA1B
SCHEMBL4242249 0.85 CCR5 (0.69) CCR5
SCHEMBL4586221 0.84 CCR5 (0.48) CCR5KCNH2CACNA1BDCUN1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed