SCHEMBL4588198

SCHEMBL4588198

Cc1ncnc(C)c1C(=O)N[C@H](C)CCN1CCC(N(Cc2ccsc2)c2ccc(OCC(=O)O)cc2)CC1

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.61
CACNA1B Q00975 1/20 0.38
FFAR1 O14842 1/20 0.37
KCNH2 Q12809 4/20 0.37
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586890 0.88 CCR5 (0.61) CCR5KCNH2OPRM1OPRD1OPRK1
SCHEMBL4587438 0.87 CCR5 (0.50) CCR5CACNA1BKCNH2
SCHEMBL4241454 0.84 CCR5 (0.85) CCR5KCNH2
SCHEMBL4586174 0.81 CCR5 (0.43) CCR5
SCHEMBL4586504 0.80 CCR5 (0.56) CCR5CACNA1BOPRM1
SCHEMBL4586351 0.79 CCR5 (0.51) CCR5CACNA1BKCNH2
SCHEMBL4586809 0.79 CCR5 (0.50) CCR5CACNA1BKCNH2
SCHEMBL4587594 0.78 CCR5 (0.48) CCR5CACNA1BKCNH2
SCHEMBL4245260 0.78 CCR5 (0.86) CCR5KCNH2
SCHEMBL13931600 0.78 CCR5 (0.84) CCR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP claimed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP claimed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO claimed
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed