SCHEMBL4587611

SCHEMBL4587611

COc1ccc(C(=O)O)c2c(=O)c(=O)c12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
MAPT P10636 3/20 0.53
TDP1 Q9NUW8 2/20 0.53
CYP1A2 P05177 1/20 0.48
KDM4E B2RXH2 6/20 0.46
HPGD P15428 4/20 0.46
CDC25B P30305 2/20 0.46
HTT P42858 3/20 0.45
LMNA P02545 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA7 P43166 2/20 0.44
CA9 Q16790 2/20 0.44
CA14 Q9ULX7 2/20 0.44
CA4 P22748 1/20 0.44
CA6 P23280 1/20 0.44
TPMT P51580 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9100503 0.86 CYP1A2 (0.61) ALDH1A1MAPTTDP1CYP1A2KDM4E
SCHEMBL4308337 0.83 KDM4E (0.49) ALDH1A1MAPTTDP1KDM4EHPGD
SCHEMBL7984639 0.79 MAPT (0.44) ALDH1A1MAPTTDP1KDM4EHPGD
SCHEMBL4308193 0.78 CYP1A2 (0.50) ALDH1A1MAPTTDP1CYP1A2KDM4E
SCHEMBL10839866 0.76 KDM4E (0.65) ALDH1A1MAPTTDP1CYP1A2KDM4E
SCHEMBL27863080 0.76 CDC25B (0.61) ALDH1A1MAPTTDP1KDM4EHPGD
SCHEMBL1203086 0.74 ALDH1A1 (0.59) ALDH1A1MAPTTDP1KDM4EHPGD
SCHEMBL7845050 0.74 CYP1A2 (0.54) ALDH1A1MAPTTDP1CYP1A2KDM4E
SCHEMBL3189109 0.72 MAPT (0.72) ALDH1A1MAPTTDP1KDM4EHPGD
SCHEMBL102827 0.72 MAPT (0.72) ALDH1A1MAPTTDP1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973405-A2 HYDROXYALKYLARYLAMIDE DERIVATIVES Merck & Co., Inc. (US) 2008-10-01 EP disclosed
WO-2007087130-A2 HYDROXYALKYLARYLAMIDE DERIVATIVES MERCK & CO., INC. (US) 2007-08-02 WO disclosed