SCHEMBL4590239

SCHEMBL4590239

Cc1ccc(-c2[c]ccs2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 9/20 0.38
NPC1 O15118 8/20 0.38
ALDH1A1 P00352 3/20 0.38
NFKB1 P19838 3/20 0.38
NFKB2 Q00653 3/20 0.38
RELA Q04206 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
MAPK1 P28482 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CASP3 P42574 2/20 0.36
ACHE P22303 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
IDO1 P14902 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3790001 0.78 CYP3A4 (0.42) RAB9ANPC1ALDH1A1SMN1; SMN2LMNA
SCHEMBL4591209 0.78 ALDH1A1 (0.36) RAB9ANPC1ALDH1A1SMN1; SMN2LMNA
SCHEMBL15546923 0.78 APP (0.44) RAB9ANPC1ALDH1A1NFKB1NFKB2
SCHEMBL27839281 0.76 ACHE (0.39) RAB9ANPC1ALDH1A1SMN1; SMN2ACHE
SCHEMBL28134941 0.74 MMP3 (0.41) ALDH1A1LMNAGAAKDM4ENOTUM
SCHEMBL6069115 0.72 TSHR (0.44) RAB9ANPC1ALDH1A1SMN1; SMN2TP53
SCHEMBL197731 0.63 ACHE (0.73) ALDH1A1LMNAACHETDP1IDO1
SCHEMBL3287696 0.63 ACHE (0.73) ALDH1A1LMNAACHETDP1IDO1
SCHEMBL18661495 0.63 ACHE (0.73) ALDH1A1LMNAACHETDP1IDO1
SCHEMBL3860 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1909775-A2 FORMULATION OF RADIOPROTECTIVE ALPHA, BETA UNSATURATED ARYL SULFONES Onconova Therapeutics, Inc. (US) 2008-04-16 EP disclosed
WO-2007016201-A2 FORMULATION OF RADIOPROTECTIVE α, β UNSATURATED ARYL SULFONES ONCONOVA THERAPEUTICS, INC. (US) 2007-02-08 WO disclosed