SCHEMBL4590686

SCHEMBL4590686

C[C](C)Cc1nc2ccc(N)cc2s1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.56
KEAP1 Q14145 1/20 0.51
MAPT P10636 10/20 0.49
GAA P10253 5/20 0.49
ALDH1A1 P00352 4/20 0.49
NPC1 O15118 4/20 0.49
RAB9A P51151 4/20 0.49
KDM4E B2RXH2 3/20 0.49
GLA P06280 3/20 0.49
HPGD P15428 3/20 0.49
TP53 P04637 2/20 0.49
PKM P14618 2/20 0.49
POLB P06746 1/20 0.49
PTBP1 P26599 1/20 0.49
CASP1 P29466 1/20 0.49
CASP7 P55210 1/20 0.49
HSD17B10 Q99714 1/20 0.49
THRB P10828 1/20 0.48
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22130286 0.83 SMN1; SMN2 (0.50) SMN1; SMN2KEAP1MAPTGAAALDH1A1
SCHEMBL10830079 0.83 SMN1; SMN2 (0.50) SMN1; SMN2KEAP1MAPTGAAALDH1A1
SCHEMBL30626914 0.81 NPC1 (0.63) SMN1; SMN2KEAP1MAPTGAAALDH1A1
SCHEMBL10047756 0.81 NPC1 (0.63) SMN1; SMN2KEAP1MAPTGAAALDH1A1
SCHEMBL20357506 0.81 SMN1; SMN2 (0.49) SMN1; SMN2KEAP1MAPTGAAALDH1A1
SCHEMBL27770393 0.81 RAB9A (0.45) SMN1; SMN2MAPTGAAALDH1A1NPC1
SCHEMBL3251161 0.80 UBE2T (0.59) SMN1; SMN2KEAP1MAPTGAAALDH1A1
SCHEMBL659302 0.77 SMN1; SMN2 (0.56) SMN1; SMN2KEAP1MAPTGAAALDH1A1
SCHEMBL27462967 0.76 MAPT (0.61) SMN1; SMN2MAPTGAAALDH1A1NPC1
SCHEMBL3203121 0.75 SMN1; SMN2 (0.53) SMN1; SMN2KEAP1MAPTGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1885719-A1 2,5- AND 2,6-DISUBSTITUTED BENZAZOLE DERIVATIVES USEFUL AS PROTEIN KINASE INHIBITORS 4SC AG (DE) 2008-02-13 EP disclosed
WO-2006066795-A1 2,5- AND 2,6-DISUBSTITUTED BENZAZOLE DERIVATIVES USEFUL AS PROTEIN KINASE INHIBITORS 4SC AG (DE) 2006-06-29 WO disclosed