SCHEMBL4590930

SCHEMBL4590930

Cc1nc(-c2ccc(C(F)(F)F)cc2C#N)[nH]c1CN(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.40
FEN1 P39748 1/20 0.40
XDH P47989 2/20 0.38
PDE2A O00408 2/20 0.36
PTGES O14684 1/20 0.35
RAF1 P04049 1/20 0.35
BRAF P15056 1/20 0.35
PIM1 P11309 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
DGAT1 O75907 2/20 0.34
SOAT1 P35610 1/20 0.34
KCNH2 Q12809 1/20 0.34
DHODH Q02127 1/20 0.33
NMT1 P30419 1/20 0.33
IDH1 O75874 1/20 0.33
CTSK P43235 1/20 0.33
LRRK2 Q5S007 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4591152 0.86 NMT1 (0.43) DHODHNMT1LRRK2
SCHEMBL4591433 0.84 POLB (0.35) PDE2APTGESDHODHNMT1LRRK2
SCHEMBL4591509 0.84 XDH (0.40) XDHPIM1PIM2DHODHCTSK
SCHEMBL4591714 0.82 KDM4E (0.39) XDHPDE2APTGESIDH1LRRK2
SCHEMBL4592213 0.82 PTGES (0.42) PTGESPIM1PIM2NMT1LRRK2
SCHEMBL4591409 0.82 LRRK2 (0.34) PTGESNMT1IDH1LRRK2
SCHEMBL4591465 0.81 KDM4E (0.40) XDHPDE2A
SCHEMBL4591626 0.80 PTGES (0.41) PTGESNMT1LRRK2CYP1A2CYP2C9
SCHEMBL5181453 0.78 VCAM1 (0.40) DHODHRECQL
SCHEMBL4592615 0.74 ALOX5AP (0.45) ALOX5APFEN1XDHPDE2APTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937688-A1 IMIDAZO BENZODIAZEPINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-07-02 EP disclosed
WO-2007042421-A1 IMIDAZO BENZODIAZEPINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-04-19 WO disclosed