SCHEMBL4590966

SCHEMBL4590966

Brc1ccc(-c2[c]nccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
MAPK1 P28482 1/20 0.39
NPC1 O15118 4/20 0.33
RAB9A P51151 4/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
CYP2A6 P11509 1/20 0.33
CYP19A1 P11511 1/20 0.33
NR1H4 Q96RI1 1/20 0.32
MAOB P27338 1/20 0.32
GAA P10253 2/20 0.31
KDM4E B2RXH2 1/20 0.31
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4590846 0.79 MAPK14 (0.35) ALDH1A1NPC1RAB9ACYP19A1MAPT
SCHEMBL2412002 0.79 NOTUM (0.39) NPC1RAB9ACYP2A6CYP19A1GAA
SCHEMBL5797199 0.78 MAPT (0.43) ALDH1A1NPC1RAB9ASMN1; SMN2CYP2A6
SCHEMBL4909130 0.77
SCHEMBL5887656 0.75 MAPT (0.47) ALDH1A1NPC1RAB9ASMN1; SMN2TSHR
SCHEMBL5066564 0.75 CLK4 (0.48) ALDH1A1NPC1RAB9ASMN1; SMN2CYP11B1
SCHEMBL4801302 0.73 LTA4H (0.45) ALDH1A1NPC1RAB9ACYP11B1CYP11B2
SCHEMBL4489657 0.71 CYP2A6 (0.56) ALDH1A1SMN1; SMN2CYP11B2CYP2A6KDM4E
SCHEMBL5543084 0.71 KMO (0.38)
SCHEMBL4806685 0.71 CYP11B1 (0.49) ALDH1A1NPC1RAB9ASMN1; SMN2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1909775-A2 FORMULATION OF RADIOPROTECTIVE ALPHA, BETA UNSATURATED ARYL SULFONES Onconova Therapeutics, Inc. (US) 2008-04-16 EP disclosed
WO-2007016201-A2 FORMULATION OF RADIOPROTECTIVE α, β UNSATURATED ARYL SULFONES ONCONOVA THERAPEUTICS, INC. (US) 2007-02-08 WO disclosed
EP-0711290-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1996-05-15 EP disclosed
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO disclosed