SCHEMBL4591098

SCHEMBL4591098

Cc1ccccc1Nc1nc(CO)c(C)c(N2CCc3ccccc3C2C)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.39
MAP4K1 Q92918 2/20 0.35
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
LMNA P02545 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
PKM P14618 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
NPSR1 Q6W5P4 2/20 0.33
KMT2A Q03164 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
NTSR1 P30989 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6968201 0.99 GBA1 (0.38) GBA1MAP4K1CCNA2CDK2CDK5
Hydrochloric Acid SCHEMBL6994237 0.90 NPC1 (0.35) GBA1MAP4K1CCNA2CDK2CDK5
Hydrochloric Acid SCHEMBL6962670 0.90 MAP4K1 (0.35) GBA1MAP4K1CCNA2CDK2CDK5
Hydrochloric Acid SCHEMBL6956801 0.87 ADRA2A (0.38) GBA1LMNANPSR1KMT2AKDM4E
SCHEMBL6990980 0.87 CCNA2 (0.37) GBA1MAP4K1CCNA2CDK2CDK5
Hydrochloric Acid SCHEMBL6990604 0.86 SMN1; SMN2 (0.38) GBA1MAP4K1CCNA2CDK2CDK5
Hydrochloric Acid SCHEMBL6993455 0.86 SMN1; SMN2 (0.38) GBA1MAP4K1CCNA2CDK2CDK5
Hydrochloric Acid SCHEMBL6999558 0.86 SMN1; SMN2 (0.38) GBA1MAP4K1CCNA2CDK2CDK5
SCHEMBL4591366 0.85 KCNH3 (0.37) LMNAKMT2AKDM4ETSHRMAPK1
Hydrochloric Acid SCHEMBL6968110 0.84 KCNH3 (0.39) LMNAKMT2AKDM4ETSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879891-A1 MUTUAL PRODRUG COMPOUNDS FOR USE AS ANTIINFLAMMATORY AGENTS WITH GASTROINTESTINAL PROTECTIVE ACTIVITY Nycomed GmbH (DE) 2008-01-23 EP claimed
WO-2006117315-A1 MUTUAL PRODRUG COMPOUNDS FOR USE AS ANTIINFLAMMATORY AGENTS WITH GASTROINTESTINAL PROTECCTIVE ACTIVITY NYCOMED GMBH (DE) 2006-11-09 WO claimed