SCHEMBL21546534

SCHEMBL21546534

C=CCc1cc(Cl)c(Cl)cc1N

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.40
GABRA1 P14867 4/20 0.35
GABRB2 P47870 4/20 0.35
CD44 P16070 1/20 0.33
PTGDR Q13258 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
HTR2A P28223 2/20 0.31
HTR2C P28335 2/20 0.31
HTR2B P41595 2/20 0.31
POLB P06746 1/20 0.31
CYP3A4 P08684 2/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6423969 0.84 GABRA1 (0.41) GAAGABRA1GABRB2POLBCYP3A4
SCHEMBL3262914 0.81 GABRA1 (0.40) GAAGABRA1GABRB2POLBCYP3A4
SCHEMBL4591472 0.78 GAA (0.40) GAACD44CYP3A4TSHR
SCHEMBL21546530 0.75 PTGDR (0.47) GABRA1GABRB2PTGDRPTGDR2POLB
SCHEMBL20819282 0.72 CYP3A4 (0.48) GAAGABRA1GABRB2PTGDRPTGDR2
SCHEMBL11196023 0.72 GABRA1 (0.32) GABRA1GABRB2HTR2CHTR2BPOLB
SCHEMBL27895858 0.72 GAA (0.48) GAACD44CYP3A4TSHR
SCHEMBL11766536 0.72 GABRA1 (0.40) GAAGABRA1GABRB2PTGDRPTGDR2
SCHEMBL1772134 0.71 GABRA1 (0.41) GAAGABRA1GABRB2POLBCYP3A4
SCHEMBL4633136 0.71 GABRA1 (0.36) GAAGABRA1GABRB2PTGDRPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3578176-A1 NON-PLATINUM-BASED ANTI-CANCER COMPOUNDS FOR USE IN TARGETED CHEMOTHERAPY Lu, Qing-Bin (CA) 2019-12-11 EP disclosed
EP-3055287-B1 NON-PLATINUM-BASED ANTI-CANCER COMPOUNDS FOR USE IN TARGETED CHEMOTHERAPY LU QING BIN (CA) 2019-11-06 EP disclosed