SCHEMBL4592034

SCHEMBL4592034

FC(F)(F)c1cccc(-c2ccc(CCl)cn2)c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 5/20 0.53
MAOB P27338 5/20 0.53
CYP11B1 P15538 1/20 0.51
CYP11B2 P19099 1/20 0.51
IDO1 P14902 1/20 0.49
GRIN1 Q05586 5/20 0.45
GRIN2B Q13224 5/20 0.45
SCN2A Q99250 1/20 0.44
MAOA P21397 2/20 0.44
KDR P35968 1/20 0.44
TEK Q02763 1/20 0.44
KMO O15229 1/20 0.44
HRH1 P35367 1/20 0.44
HRH4 Q9H3N8 1/20 0.44
CTSS P25774 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4591309 0.85 MAOB (0.53) KDM1AMAOBCYP11B1CYP11B2IDO1
SCHEMBL21093319 0.83 NPC1 (0.54) KDM1AMAOBCYP11B1CYP11B2IDO1
SCHEMBL5515167 0.82 CYP11B1 (0.45) KDM1AMAOBCYP11B1CYP11B2IDO1
SCHEMBL1550000 0.81 CYP11B1 (0.49) KDM1AMAOBCYP11B1CYP11B2KDR
SCHEMBL1416558 0.81 KDM1A (0.61) KDM1AMAOBIDO1SCN2AMAOA
Hydrochloric Acid SCHEMBL31375590 0.80 CYP11B1 (0.48) KDM1AMAOBCYP11B1CYP11B2IDO1
SCHEMBL6240438 0.80 KDM1A (0.57) KDM1AMAOBIDO1SCN2AMAOA
SCHEMBL6236148 0.78 KDM1A (0.58) KDM1AMAOBIDO1SCN2AMAOA
SCHEMBL27174439 0.78 MAOB (0.64) KDM1AMAOBGRIN1GRIN2BKDR
SCHEMBL6235013 0.77 KDM1A (0.57) KDM1AMAOBIDO1SCN2AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7429605-B2 Phenylpyridine derivatives HOFFMANN-LA ROCHE INC. (US) 2008-09-30 US disclosed
CN-101213186-A Phenylpyridine derivatives, their manufacture and use as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2008-07-02 CN disclosed
EP-1912969-A1 PHENYLPYRIDINE DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2008-04-23 EP disclosed
WO-2007017169-A1 PHENYLPYRIDINE DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2007-02-15 WO disclosed
US-20070032530-A1 Phenylpyridine derivatives HOFFMANN-LA ROCHE INC. 2007-02-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070032530-A1 Phenylpyridine derivatives CYP3A5, QDPR, DPYD KDM1A 2483/4885MAOB 211/4885CYP11B1 127/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.