SCHEMBL459209

SCHEMBL459209

COn1c(-c2cccnc2)nc2cc(S(C)(=O)=O)ccc21

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.48
PTGS1 P23219 3/20 0.45
CYP11B1 P15538 4/20 0.42
CYP11B2 P19099 4/20 0.42
ALOX5AP P20292 1/20 0.41
USP2 O75604 1/20 0.41
HTT P42858 1/20 0.41
NCOA1 Q15788 1/20 0.41
NCOA3 Q9Y6Q9 1/20 0.41
NPC1 O15118 1/20 0.41
CASP3 P42574 1/20 0.41
RAB9A P51151 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
SENP6 Q9GZR1 1/20 0.41
LRRK2 Q5S007 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896747 0.87 PTGS2 (0.46) PTGS2PTGS1CYP11B1CYP11B2ALOX5AP
SCHEMBL17883781 0.84 PTGS2 (0.57) PTGS2PTGS1CYP11B1CYP11B2NPC1
SCHEMBL17896745 0.83 PTGS2 (0.51) PTGS2PTGS1CYP11B1CYP11B2ALOX5AP
SCHEMBL10175792 0.81 CYP11B2 (0.46) CYP11B1CYP11B2ALOX5APUSP2HTT
SCHEMBL10175134 0.81 CYP11B1 (0.59) PTGS2PTGS1CYP11B1CYP11B2HTT
SCHEMBL10175131 0.81 USP2 (0.65) PTGS2PTGS1CYP11B1CYP11B2ALOX5AP
SCHEMBL460487 0.80 CYP11B2 (0.41) CYP11B1CYP11B2ALOX5APUSP2HTT
SCHEMBL458763 0.80 CYP11B2 (0.43) CYP11B1CYP11B2ALOX5APUSP2HTT
SCHEMBL10175133 0.79 CYP11B2 (0.68) PTGS2CYP11B1CYP11B2
SCHEMBL17896649 0.71 PTGS2 (0.58) PTGS2PTGS1CYP11B1CYP11B2ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
EP-2595482-A1 ALDOSTERONE SYNTHASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-05-29 EP disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed