SCHEMBL4592149

SCHEMBL4592149

CN(C)CC(=C=O)c1ccc(C(F)(F)F)cc1F

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CYP11B1 P15538 2/20 0.41
CYP11B2 P19099 2/20 0.41
PDE2A O00408 2/20 0.39
KDM4E B2RXH2 2/20 0.39
HTT P42858 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
PDK2 Q15119 2/20 0.38
CES2 O00748 1/20 0.37
POLQ O75417 2/20 0.37
NTRK1 P04629 2/20 0.37
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CFTR P13569 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5772527 0.77 LSS (0.44) CES2
SCHEMBL5771539 0.75 CES2 (0.50) CES2ALDH1A1
SCHEMBL5772127 0.72 LMNA (0.42) GAASMN1; SMN2L3MBTL1POLQALDH1A1
SCHEMBL29499840 0.70 GAA (0.58) GAASMN1; SMN2L3MBTL1CYP11B1CYP11B2
SCHEMBL1350804 0.70 GAA (0.58) GAASMN1; SMN2L3MBTL1CYP11B1CYP11B2
SCHEMBL694388 0.69 CFTR (0.69) GAASMN1; SMN2L3MBTL1CYP11B1CYP11B2
SCHEMBL2075208 0.69 GAA (0.54) GAASMN1; SMN2L3MBTL1CYP11B1CYP11B2
SCHEMBL28188798 0.69 GAA (0.57) GAASMN1; SMN2L3MBTL1CYP11B1CYP11B2
SCHEMBL16647662 0.69 MRGPRX4 (0.51) GAASMN1; SMN2L3MBTL1PDE2AKDM4E
SCHEMBL26057003 0.68 GAA (0.56) GAASMN1; SMN2L3MBTL1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912969-A1 PHENYLPYRIDINE DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2008-04-23 EP disclosed
WO-2007017169-A1 PHENYLPYRIDINE DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2007-02-15 WO disclosed