SCHEMBL5771539

SCHEMBL5771539

CN(C)CC(=C=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.50
ALDH1A1 P00352 2/20 0.49
POLB P06746 1/20 0.46
NPSR1 Q6W5P4 1/20 0.44
LMNA P02545 1/20 0.44
SRD5A2 P31213 1/20 0.43
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
PTGS1 P23219 1/20 0.42
OPRM1 P35372 1/20 0.41
OPRL1 P41146 1/20 0.41
P2RX1 P51575 1/20 0.41
TP53 P04637 1/20 0.41
TP53BP1 Q12888 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5772527 0.81 LSS (0.44) CES2SRD5A2MEN1KMT2A
SCHEMBL5489563 0.77 HPGD (0.45) ALDH1A1POLBTP53
SCHEMBL4592149 0.75 GAA (0.50) CES2ALDH1A1
SCHEMBL7411270 0.74 CES2 (0.59) CES2ALDH1A1POLBNPSR1LMNA
SCHEMBL5779568 0.72 BCHE (0.43)
SCHEMBL7899079 0.72 CES2 (0.56) CES2ALDH1A1POLBNPSR1SRD5A2
SCHEMBL3876454 0.71 CES2 (0.65) CES2ALDH1A1POLBNPSR1LMNA
SCHEMBL20870672 0.71 CES2 (0.65) CES2ALDH1A1POLBNPSR1LMNA
SCHEMBL4245460 0.71 OPRM1 (0.64) CES2ALDH1A1POLBNPSR1LMNA
Hydrochloric Acid SCHEMBL4420249 0.71 CES2 (0.54) CES2ALDH1A1POLBNPSR1SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1648896-A1 7-SUBSTITUTED 3-NITRO-PYRAZOLO [1,5-A] PYRIMIDINES FERRER INTERNACIONAL, S.A. (ES) 2006-04-26 EP disclosed
WO-2005014596-A1 7-SUBSTITUTED 3-NITRO-PYRAZOLO `1,5-A! PYRIMIDINES FERRER INTERNACIONAL, S.A. (ES) 2005-02-17 WO disclosed