SCHEMBL4592248

SCHEMBL4592248

Nc1c(CC=O)ccc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
HSD17B10 Q99714 4/20 0.41
HPGD P15428 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
GLA P06280 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41
CYP1B1 Q16678 2/20 0.40
CYP1A1 P04798 1/20 0.40
TSHR P16473 2/20 0.39
CYP2A6 P11509 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
NCEH1 Q6PIU2 1/20 0.38
ERN1 O75460 1/20 0.38
CYP3A4 P08684 1/20 0.38
KEAP1 Q14145 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2161442 0.81 ALDH1A1 (0.41) ALDH1A1HSD17B10HPGDKDM4EMEN1
Formic Acid SCHEMBL27532730 0.79 NCEH1 (0.43) ALDH1A1HSD17B10HPGDKDM4EMEN1
SCHEMBL1556062 0.79 NCEH1 (0.45) ALDH1A1HSD17B10HPGDKDM4EMEN1
SCHEMBL31148944 0.78 POLB (0.46) ALDH1A1HSD17B10HPGDPOLBMAPT
SCHEMBL11746597 0.78 CYP2A6 (0.48) ALDH1A1HSD17B10TSHRCYP2A6TDP1
SCHEMBL2012510 0.78 PTPN22 (0.48)
SCHEMBL2016155 0.78 POLB (0.46) ALDH1A1HSD17B10HPGDPOLBMAPT
SCHEMBL720557 0.76 CYP1A2 (0.52) ALDH1A1HPGDMEN1MAPTKMT2A
SCHEMBL2891376 0.76 ALDH1A1 (0.46) ALDH1A1HSD17B10HPGDKDM4EMEN1
SCHEMBL23663727 0.75 ALDH1A1 (0.44) ALDH1A1HSD17B10HPGDKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888538-A1 (3,4-DIHYDRO-QUINAZOLIN-2-YL)-(2-ARYLOXY-ETHYL)-AMINES HAVING AN ACTIVITY ON THE 5-HT RECEPTOR F. Hoffmann-Roche AG (CH) 2008-02-20 EP disclosed
WO-2006117305-A1 (3,4-DIHYDRO-QUINAZOLIN-2-YL)-(2-ARYLOXY-ETHYL)-AMINES HAVING AN ACTIVITY ON THE 5-HT RECEPTOR F. HOFFMANN-LA ROCHE AG (CH) 2006-11-09 WO disclosed