SCHEMBL4593078

SCHEMBL4593078

Cc1ccc(-c2cccc(N)c2)cc1.Cc1ccc(-c2cccc([N+](=O)[O-])c2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.62
TSHR P16473 2/20 0.53
ACHE P22303 2/20 0.53
GAA P10253 2/20 0.50
MAPT P10636 2/20 0.50
NPC1 O15118 1/20 0.50
HPGD P15428 1/20 0.50
CASP3 P42574 1/20 0.50
HTT P42858 1/20 0.50
RAB9A P51151 1/20 0.50
SENP7 Q9BQF6 1/20 0.50
NFE2L2 Q16236 1/20 0.50
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
LMNA P02545 2/20 0.47
PGR P06401 3/20 0.47
MMP2 P08253 1/20 0.47
MMP9 P14780 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1036939 0.91 TSHR (0.63) ALDH1A1TSHRACHEGAAMAPT
SCHEMBL2026676 0.89 ALDH1A1 (0.78) ALDH1A1TSHRACHEGAAMAPT
SCHEMBL30469275 0.89 ALDH1A1 (0.78) ALDH1A1TSHRACHEGAAMAPT
Water SCHEMBL29134001 0.87 ALDH1A1 (0.75) ALDH1A1TSHRACHEGAAMAPT
SCHEMBL30360587 0.84 ALDH1A1 (0.63) ALDH1A1TSHRACHEGAAMAPT
SCHEMBL7142305 0.84 ALDH1A1 (0.63) ALDH1A1TSHRACHEGAAMAPT
SCHEMBL26673982 0.84 ALDH1A1 (0.63) ALDH1A1TSHRMAPTNPC1RAB9A
SCHEMBL23542887 0.82 MAOA (0.67) ALDH1A1ACHEMAPTNPC1HPGD
SCHEMBL1040119 0.82 MAOA (0.67) ALDH1A1ACHEMAPTNPC1HPGD
Dinitrophenylene SCHEMBL27461706 0.80 ALDH1A1 (0.63) ALDH1A1TSHRACHEGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1948616-A1 2-(BENZIMIDAZOL-1-YL)-ACETAMIDE BIARYL DERIVATIVES AND THEIR USE AS INHIBITORS OF THE TRPV1 RECEPTOR N.V. Organon (NL) 2008-07-30 EP disclosed
WO-2007054480-A1 2-(BENZIMIDAZOL-1-YL)-ACETAMIDE BIARYL DERIVATIVES AND THEIR USE AS INHIBITORS OF THE TRPV1 RECEPTOR N.V. ORGANON (NL) 2007-05-18 WO disclosed