SCHEMBL4593174

SCHEMBL4593174

CC(=O)CCC(c1cc(F)cc(F)c1)N(C)C

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
CHRNB2 P17787 2/20 0.35
CHRNB4 P30926 2/20 0.35
CHRNA3 P32297 2/20 0.35
CHRNA4 P43681 2/20 0.35
OPRM1 P35372 9/20 0.34
OPRL1 P41146 8/20 0.34
ACKR3 P25106 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4593455 0.75 CES2 (0.41) CES2CES1OPRM1OPRL1ACKR3
SCHEMBL6421263 0.70 CES2 (0.32) CES2CES1OPRM1OPRL1
SCHEMBL6012109 0.69 CES2 (0.41) CES2CES1OPRM1OPRL1
SCHEMBL12861273 0.68 OPRM1 (0.52) CES2CES1OPRM1OPRL1
SCHEMBL7496510 0.66 OPRM1 (0.43) OPRM1
SCHEMBL23085208 0.65 ALDH1A1 (0.52) CES2CES1
SCHEMBL8109949 0.65 CACNA1B (0.50) OPRM1
SCHEMBL22608928 0.63 CES2 (0.36) CES2CES1
SCHEMBL8141135 0.63 HTT (0.42)
SCHEMBL14537114 0.62 CES2 (0.61) CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1898914-A1 QUINOLINE DERIVATIVES AS ANTIBACTERIAL AGENTS JANSSEN PHARMACEUTICA N.V. (BE) 2008-03-19 EP disclosed
WO-2007000435-A1 QUINOLINE DERIVATIVES AS ANTIBACTERIAL AGENTS JANSSEN PHARMACEUTICA N.V. (BE) 2007-01-04 WO disclosed