SCHEMBL4593306

SCHEMBL4593306

FC(F)(F)c1cccc(Nn2cccn2)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.52
POLB P06746 1/20 0.52
KIF11 P52732 1/20 0.49
IDH2 P48735 2/20 0.46
AURKA O14965 1/20 0.44
MAPT P10636 4/20 0.44
ALDH1A1 P00352 2/20 0.44
GAA P10253 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
MEN1 O00255 1/20 0.43
HTT P42858 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.42
KDM4E B2RXH2 1/20 0.42
RAPGEF4 Q8WZA2 1/20 0.42
IDO1 P14902 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28781470 0.81 NOTUM (0.54) LMNAPOLBKIF11IDH2AURKA
SCHEMBL27641960 0.75 KIF11 (0.50) LMNAPOLBKIF11IDH2AURKA
SCHEMBL825684 0.73 CYP1A2 (0.38) LMNAALDH1A1GAATDP1L3MBTL1
SCHEMBL29748950 0.70 MAPT (0.58) KIF11IDH2MAPTALDH1A1GAA
SCHEMBL2925587 0.70 MAPT (0.58) KIF11IDH2MAPTALDH1A1GAA
SCHEMBL394991 0.70 KIF11 (0.70) LMNAKIF11IDH2AURKAMAPT
SCHEMBL11286034 0.70 NOTUM (0.64) LMNAMAPTALDH1A1HTTRAB9A
SCHEMBL1807928 0.70 MEN1 (0.56) LMNAPOLBIDH2MAPTALDH1A1
SCHEMBL30402678 0.70 NOTUM (0.64) LMNAMAPTALDH1A1HTTRAB9A
SCHEMBL30047371 0.70 HTT (0.55) LMNAPOLBMAPTALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910347-A2 MACROCYLIC INHIBITORS OF HEPATITIS C VIRUS MEDIVIR AB (SE) 2008-04-16 EP disclosed
WO-2007017144-A2 MACROCYLIC INHIBITORS OF HEPATITIS C VIRUS MEDIVIR AB (SE) 2007-02-15 WO disclosed