SCHEMBL4593462

SCHEMBL4593462

COC(=O)c1ccc2oc(N(Cc3cc(OC(C)C)cc(OC(C)C)c3)C3CCNCC3)nc2c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.40
CMKLR1 Q99788 1/20 0.39
ALOX5AP P20292 1/20 0.37
FEN1 P39748 1/20 0.37
MBTPS1 Q14703 1/20 0.37
HDAC6 Q9UBN7 3/20 0.37
MAPT P10636 5/20 0.36
THRB P10828 2/20 0.36
IDH1 O75874 1/20 0.36
ELANE P08246 1/20 0.35
SSTR5 P35346 1/20 0.35
HTR2A P28223 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TP53 P04637 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4594611 0.93 TP53 (0.38) RAB9ANPC1MBTPS1MAPTTHRB
SCHEMBL4594412 0.92 HDAC6 (0.38) RAB9ANPC1MBTPS1HDAC6MAPT
SCHEMBL4593931 0.88 KDM4E (0.40) RAB9ANPC1CMKLR1MBTPS1MAPT
SCHEMBL4594697 0.86 GAA (0.41) IDH1HTR2A
SCHEMBL4593295 0.85 TP53 (0.39) MBTPS1SSTR5HTR2ATP53KMT2A
SCHEMBL4593394 0.84 SLC6A2 (0.36) MBTPS1SSTR5HTR2A
SCHEMBL4594214 0.84 MAPK1 (0.36) MBTPS1SSTR5HTR2ASMN1; SMN2KMT2A
SCHEMBL4593207 0.82 SSTR5 (0.36) MBTPS1SSTR5HTR2ASMN1; SMN2
SCHEMBL4594514 0.82 SSTR5 (0.46) RAB9ANPC1CMKLR1ALOX5APFEN1
SCHEMBL4593460 0.82 SSTR5 (0.47) RAB9ANPC1CMKLR1ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924579-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-05-28 EP claimed
WO-2007025897-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-03-08 WO claimed
EP-1924579-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-05-28 EP disclosed
WO-2007025897-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-03-08 WO disclosed