SCHEMBL4594611

SCHEMBL4594611

COC(=O)c1ccc2nc(N(Cc3cc(OC(C)C)cc(OC(C)C)c3)C3CCNCC3)oc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.38
MBTPS1 Q14703 1/20 0.37
CTSL P07711 1/20 0.36
CTSS P25774 1/20 0.36
MAPT P10636 5/20 0.36
THRB P10828 1/20 0.36
ELANE P08246 1/20 0.35
SSTR5 P35346 1/20 0.35
HTR2A P28223 1/20 0.35
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
NFKB1 P19838 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
ATM Q13315 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4593462 0.93 RAB9A (0.40) TP53MBTPS1MAPTTHRBELANE
SCHEMBL4593295 0.92 TP53 (0.39) TP53MBTPS1SSTR5HTR2AKDM4E
SCHEMBL4594412 0.85 HDAC6 (0.38) TP53MBTPS1MAPTTHRBSSTR5
SCHEMBL4593931 0.83 KDM4E (0.40) MBTPS1MAPTSSTR5HTR2AKDM4E
SCHEMBL4593756 0.82 SSTR5 (0.47) TP53CTSLCTSSMAPTSSTR5
SCHEMBL4594089 0.82 SSTR5 (0.39) TP53MAPTSSTR5KDM4ENPC1
SCHEMBL4593912 0.82 SSTR5 (0.41) TP53MAPTSSTR5KDM4ENPC1
SCHEMBL4593748 0.82 SSTR5 (0.41) TP53MAPTSSTR5NPC1RAB9A
SCHEMBL4594697 0.81 GAA (0.41) HTR2AKDM4EIDH1PPARGPPARD
SCHEMBL4593487 0.80 TRPV1 (0.38) TP53MBTPS1MAPTTHRBHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924579-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-05-28 EP disclosed
WO-2007025897-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-03-08 WO disclosed