SCHEMBL4594412

SCHEMBL4594412

CC(C)Oc1cc(CN(c2nc3cc(C(=O)O)ccc3o2)C2CCNCC2)cc(OC(C)C)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.38
MBTPS1 Q14703 2/20 0.38
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TP53 P04637 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
PTGER1 P34995 1/20 0.37
PTGER3 P43115 1/20 0.37
PTGER2 P43116 1/20 0.37
KMT2A Q03164 1/20 0.37
PTGDR Q13258 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PPARD Q03181 6/20 0.36
PPARA Q07869 6/20 0.36
PPARG P37231 4/20 0.36
HTR2A P28223 1/20 0.36
MAPT P10636 1/20 0.35
SSTR5 P35346 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4593295 0.93 TP53 (0.39) MBTPS1KDM4EMEN1ALDH1A1TP53
SCHEMBL4593462 0.92 RAB9A (0.40) HDAC6MBTPS1TP53KMT2AHTR2A
SCHEMBL4594697 0.89 GAA (0.41) KDM4EPPARDPPARAPPARGHTR2A
SCHEMBL4593931 0.86 KDM4E (0.40) MBTPS1KDM4EALDH1A1PPARDPPARA
SCHEMBL4593394 0.85 SLC6A2 (0.36) MBTPS1PPARDPPARAPPARGHTR2A
SCHEMBL4594214 0.85 MAPK1 (0.36) MBTPS1KDM4EMEN1ALDH1A1KMT2A
SCHEMBL4594611 0.85 TP53 (0.38) MBTPS1KDM4EALDH1A1TP53HPGD
SCHEMBL4593207 0.84 SSTR5 (0.36) MBTPS1ALDH1A1PPARDPPARAPPARG
SCHEMBL4594418 0.83 PPARD (0.37) PPARDPPARAPPARGHTR2ASSTR5
SCHEMBL4594500 0.83 PPARD (0.35) PPARDPPARAPPARGSSTR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924579-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-05-28 EP claimed
WO-2007025897-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-03-08 WO claimed
EP-1924579-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-05-28 EP disclosed
WO-2007025897-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-03-08 WO disclosed