SCHEMBL4593507

SCHEMBL4593507

CC(C)=CCC(=CCN[C@@H](CS)C(=O)O)CCc1ccc(-c2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ICMT O60725 2/20 0.51
FFAR1 O14842 2/20 0.41
MMP12 P39900 1/20 0.40
MME P08473 9/20 0.39
ACE P12821 8/20 0.39
ACE2 Q9BYF1 8/20 0.39
CPA1 P15085 6/20 0.39
TRPV1 Q8NER1 1/20 0.38
FFAR4 Q5NUL3 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4592994 0.85 FFAR1 (0.46) ICMTFFAR1MMP12MMEACE
SCHEMBL13129949 0.76 FFAR1 (0.46) ICMTFFAR1MMP12TRPV1FFAR4
SCHEMBL2815696 0.76 FFAR1 (0.46) ICMTFFAR1MMP12TRPV1FFAR4
SCHEMBL5445097 0.76 ICMT (0.72) ICMTACE
SCHEMBL14596300 0.76 ICMT (0.72) ICMTACE
SCHEMBL14596301 0.75 ICMT (0.46) ICMTFFAR1MMP12TRPV1FFAR4
SCHEMBL13883693 0.73 ICMT (0.51) ICMTFFAR1MMP12TRPV1FFAR4
SCHEMBL332020 0.72 MAPT (0.52) ACE
SCHEMBL388271 0.72 MAPT (0.52) ACE
SCHEMBL1762279 0.72 MAPT (0.52) ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613585-A4 COMPOUNDS AND METHODS FOR USE IN TREATING NEOPLASIA AND CANCER BASED UPON INHIBITORS OF ISOPRENYLCYSTEINE METHYLTRANSFERASE PURDUE RESEARCH FOUNDATION (US) 2008-07-23 EP disclosed
EP-1613585-A2 COMPOUNDS AND METHODS FOR USE IN TREATING NEOPLASIA AND CANCER BASED UPON INHIBITORS OF ISOPRENYLCYSTEINE METHYLTRANSFERASE PURDUE RESEARCH FOUNDATION (US) 2006-01-11 EP disclosed
WO-2004087064-A2 COMPOUNDS AND METHODS FOR USE IN TREATING NEOPLASIA AND CANCER BASED UPON INHIBITORS OF ISOPRENYLCYSTEINE METHYLTRANSFERASE PURDUE RESEARCH FOUNDATION (US) 2004-10-14 WO disclosed