Methane

Methane

SCHEMBL4593708

C.CCCCCN1C(=O)CCC1C

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.44
CHRM4 P08173 3/20 0.44
CHRM5 P08912 3/20 0.44
CHRM1 P11229 3/20 0.44
CHRM3 P20309 3/20 0.44
PTGER4 P35408 8/20 0.43
PTGER3 P43115 6/20 0.43
PTGER2 P43116 5/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
POLB P06746 1/20 0.43
FAAH O00519 2/20 0.41
MGLL Q99685 2/20 0.41
GBA1 P04062 1/20 0.41
TP53 P04637 2/20 0.39
GAA P10253 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MDM2 Q00987 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4635213 0.98 CHRM2 (0.45) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL30697351 0.96 PTGER4 (0.46) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL664648 0.96 PTGER4 (0.46) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL665342 0.96 PTGER4 (0.46) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL4329362 0.96 PTGER4 (0.46) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL4588206 0.96 PTGER4 (0.46) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL4588711 0.96 PTGER4 (0.46) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL664674 0.96 PTGER4 (0.46) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL4588299 0.96 PTGER4 (0.46) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL1869119 0.93 MEN1 (0.48) CHRM2CHRM4CHRM5CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1605934-A4 PRODUCTION OF 5-METHYL-N-(METHYL ARYL)-2-PYRROLIDONE, 5-METHYL-N-(METHYL CYCLOALKYL)-2-PYRROLIDONE AND 5-METHYL-N-ALKYL-2-PYRROLIDONE DU PONT (US) 2008-10-08 EP disclosed
EP-1606046-A4 PRODUCTION OF 5-METHYL-N-(METHYL ARYL)-2-PYRROLIDONE, 5-METHYL-N-(METHYL CYCLOALKYL)-2-PYRROLIDONE AND 5- METHYL-N-ALKYL-2-PYRROLIDONE BY REDUCTIVE AMINATION OF LEUVLINIC ACID ESTERS WITH CYANO COMPOUNDS DU PONT (US) 2008-06-25 EP disclosed
EP-1605934-A1 PRODUCTION OF 5-METHYL-N-(METHYL ARYL)-2-PYRROLIDONE, 5-METHYL-N-(METHYL CYCLOALKYL)-2-PYRROLIDONE AND 5-METHYL-N-ALKYL-2-PYRROLIDONE E.I. DUPONT DE NEMOURS AND COMPANY, Legal Patent Records Center (US) 2005-12-21 EP disclosed
EP-1606046-A2 PRODUCTION OF 5-METHYL-N-(METHYL ARYL)-2-PYRROLIDONE, 5-METHYL-N-(METHYL CYCLOALKYL)-2-PYRROLIDONE AND 5- METHYL-N-ALKYL-2-PYRROLIDONE BY REDUCTIVE AMINATION OF LEUVLINIC ACID ESTERS WITH CYANO COMPOUNDS E.I. Dupont De Nemours (US) 2005-12-21 EP disclosed
WO-2004085048-A3 PRODUCTION OF 5-METHYL-N-(METHYL ARYL)-2-PYRROLIDONE, 5-METHYL-N-(METHYL CYCLOALKYL)-2-PYRROLIDONE AND 5- METHYL-N-ALKYL-2-PYRROLIDONE BY REDUCTIVE AMINATION OF LEUVLINIC ACID ESTERS WITH CYANO COMPOUNDS DU PONT (US) 2005-09-01 WO disclosed
WO-2004084888-A1 PRODUCTION OF 5-METHYL-N-(METHYL ARYL)-2-PYRROLIDONE, 5-METHYL-N-(METHYL CYCLOALKYL)-2-PYRROLIDONE AND 5-METHYL-N-ALKYL-2-PYRROLIDONE E.I. DUPONT DE NEMOURS AND COMPANY (US) 2004-10-07 WO disclosed
WO-2004085048-A2 PRODUCTION OF 5-METHYL-N-(METHYL ARYL)-2-PYRROLIDONE, 5-METHYL-N-(METHYL CYCLOALKYL)-2-PYRROLIDONE AND 5- METHYL-N-ALKYL-2-PYRROLIDONE BY REDUCTIVE AMINATION OF LEUVLINIC ACID ESTERS WITH CYANO COMPOUNDS E.I. DUPONT DE NEMOURS AND COMPANY (US) 2004-10-07 WO disclosed