SCHEMBL4593743

SCHEMBL4593743

COc1c[c]c(C(N)=O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.52
CA2 P00918 4/20 0.52
PARP10 Q53GL7 2/20 0.52
PARP1 P09874 2/20 0.52
PARP2 Q9UGN5 1/20 0.52
PARP4 Q9UKK3 1/20 0.52
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38
MAP4K4 O95819 1/20 0.38
IKBKB O14920 1/20 0.38
KDM4E B2RXH2 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
PRNP P04156 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3956678 0.82 HPGD (0.43) CA1CA2PARP10PARP1PARP2
SCHEMBL8755333 0.82 CA1 (0.50) CA1CA2PARP10PARP1PARP2
SCHEMBL28022989 0.81 PRSS1 (0.52) CA1CA2PARP10PARP1PARP2
SCHEMBL7302208 0.81 CA1 (0.52) CA1CA2PARP10PARP1PARP2
SCHEMBL28656480 0.77 PARP10 (0.58) CA1CA2PARP10PARP2PARP4
SCHEMBL9786928 0.75 CES2 (0.51) CA1CA2CES2CES1ALDH1A1
SCHEMBL10636083 0.74 PARP1 (0.36) PARP10PARP1CES2CES1ALDH1A1
SCHEMBL7753773 0.73 TP53 (0.48) CA1CA2PARP10PARP1PARP2
SCHEMBL18554580 0.73 PARP1 (0.50) CA1CA2PARP10PARP1PARP2
SCHEMBL7304754 0.71 PARP10 (0.41) CA1CA2PARP10PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1948639-A2 NOVEL CARBOCYCLIC FUSED CYCLIC AMINES F. Hoffmann-la Roche AG (CH) 2008-07-30 EP disclosed
WO-2007054453-A2 CARBOCYCLIC FUSED CYCLIC AMINES AS INHIBITORS OF THE COAGULATION FACTOR XA F. HOFFMANN-LA ROCHE AG (CH) 2007-05-18 WO disclosed