SCHEMBL7753773

SCHEMBL7753773

COc1ccc(C(=O)N(c2c[c]c(C(N)=O)cc2)S(C)(=O)=O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 5/20 0.48
LMNA P02545 2/20 0.48
KMT2A Q03164 4/20 0.46
ALDH1A1 P00352 3/20 0.46
PARP10 Q53GL7 2/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
PARP1 P09874 1/20 0.44
PARP2 Q9UGN5 1/20 0.44
PARP4 Q9UKK3 1/20 0.44
HSP90AA1 P07900 3/20 0.42
MAPT P10636 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
THRB P10828 1/20 0.42
KDM4E B2RXH2 2/20 0.40
MEN1 O00255 1/20 0.40
HPGD P15428 1/20 0.40
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4593743 0.73 CA1 (0.52) ALDH1A1PARP10CA1CA2PARP1
SCHEMBL7753781 0.72 PARP10 (0.43) TP53LMNAKMT2AALDH1A1PARP10
SCHEMBL17292712 0.68 PARP10 (0.70) TP53LMNAKMT2AALDH1A1PARP10
SCHEMBL7736889 0.68 CES2 (0.52) TP53LMNAKMT2AALDH1A1PARP10
SCHEMBL7745401 0.67 TP53 (0.43) TP53LMNAKMT2AALDH1A1HSP90AA1
SCHEMBL2112462 0.66 KDM4E (0.59) TP53LMNAKMT2AALDH1A1PARP10
SCHEMBL10049412 0.66 CA1 (0.59) ALDH1A1PARP10CA1CA2PARP1
SCHEMBL834715 0.65 TP53 (1.00) TP53LMNAKMT2AALDH1A1HSP90AA1
SCHEMBL5830407 0.65 ALDH1A1 (0.43) KMT2AALDH1A1PARP10CA1CA2
SCHEMBL201761 0.65 PARP10 (1.00) KMT2AALDH1A1PARP10CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070055-A1 SUBSTITUTED PHENYL PYRIDAZINONES Bayer Aktiengesellschaft (DE) 2001-01-24 EP disclosed
WO-1999052878-A1 SUBSTITUTED PHENYL PYRIDAZINONES BAYER AKTIENGESELLSCHAFT (DE) 1999-10-21 WO disclosed