SCHEMBL4594705

SCHEMBL4594705

C=CCOC(=O)c1c[nH]cn1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.47
ALDH1A1 P00352 3/20 0.41
HSD17B10 Q99714 2/20 0.41
TSHR P16473 1/20 0.41
SNCA P37840 1/20 0.41
KDM4E B2RXH2 2/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38
MEN1 O00255 5/20 0.36
KMT2A Q03164 5/20 0.36
RHOA P61586 1/20 0.36
MAPT P10636 3/20 0.36
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
MAPK1 P28482 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9212743 0.79 LMNA (0.33) ALDH1A1MAPTLMNA
SCHEMBL179565 0.79 CYP1A2 (0.50) ALDH1A1HSD17B10TSHRKDM4EHPGD
SCHEMBL29158197 0.76 CYP3A4 (0.47) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL3015836 0.76 ALDH1A1 (0.44) CYP3A4ALDH1A1HSD17B10TSHRKDM4E
SCHEMBL1437231 0.76 KDM4E (0.39) ALDH1A1KDM4EMEN1KMT2ALMNA
SCHEMBL25475161 0.76 FNTA (0.33) ALDH1A1MAPTLMNA
SCHEMBL3555935 0.75
SCHEMBL1397897 0.75 CYP3A4 (0.59) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL27493011 0.75 ALDH1A1 (0.35) ALDH1A1KDM4E
SCHEMBL8055864 0.73 MEN1 (0.54) CYP3A4ALDH1A1HSD17B10TSHRSNCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070036718-A1 Radio-halogenated carboxylic ester derivatives of phenylethyl imidazole tomography/scintigraphy imaging for detection of adrenal cortical pathology, e.g. incidentaloma, adenoma, primary and metastatic cortical carcinoma; highly selective with a high rate of accumulation in adrenals; antitumor agents ZOLLE, ILSE (AT) 2007-02-15 US claimed
US-20050033060-A1 Radiolabelled phenylethyl imidazole caboxylic acid ester derivatives ZOLLE, ILSE (AT) 2005-02-10 US claimed
US-4055573-A TO 4-HYDROXYMETHYL OR ALKOXYMETHYL IMIDAZOLES SMITHKLINE CORPORATION (US) 1977-10-25 US claimed
US-20080009506-A1 Imidazole Compound MITSUBISHI TANABE PHARMA CORPORATION (JP) 2008-01-10 US disclosed
EP-0338939-A1 Histamine derivative, process for his preparation and his therapeutic application INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1989-10-25 EP disclosed
US-4322539-A BY REACTION WITH AMINOALKYLENE THIOLS ETHYL CORPORATION (US) 1982-03-30 US disclosed
US-4055573-A TO 4-HYDROXYMETHYL OR ALKOXYMETHYL IMIDAZOLES SMITHKLINE CORPORATION (US) 1977-10-25 US disclosed
US-4055573-A TO 4-HYDROXYMETHYL OR ALKOXYMETHYL IMIDAZOLES SMITHKLINE CORPORATION (US) 1977-10-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070036718-A1 Radio-halogenated carboxylic ester derivatives of phenylethyl imidazole tomography/scintigraphy imaging for detection of adrenal cortical pathology, e.g. incidentaloma, adenoma, primary and metastatic cortical carcinoma; highly selective with a high rate of accumulation in adrenals; antitumor agents CDC73, TPD52L2, NTRK1 CYP3A4 105/4885ALDH1A1 1747/4885HSD17B10 810/4885
US-20080009506-A1 Imidazole Compound KCNH2, KCNJ2, KCNH3 CYP3A4 1244/4885ALDH1A1 2945/4885HSD17B10 3428/4885
US-20050033060-A1 Radiolabelled phenylethyl imidazole caboxylic acid ester derivatives CDC73, BRDT, TEC CYP3A4 777/4885ALDH1A1 2333/4885HSD17B10 1289/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.