SCHEMBL4595012

SCHEMBL4595012

CC(=O)OOc1ccc(C(F)(F)F)cc1C#N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.45
PTPN6 P29350 1/20 0.45
PTPN11 Q06124 1/20 0.45
TAS2R14 Q9NYV8 1/20 0.45
CYP2C19 P33261 3/20 0.43
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
USP2 O75604 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
PTGDR2 Q9Y5Y4 4/20 0.41
MRGPRX4 Q96LA9 2/20 0.40
ESRRA P11474 1/20 0.40
AR P10275 3/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 2/20 0.40
RECQL P46063 1/20 0.40
ACACB O00763 1/20 0.39
SCN9A Q15858 1/20 0.38
BACE1 P56817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4595015 0.85 CYP2C19 (0.56) PTPN1PTPN6PTPN11TAS2R14CYP2C19
SCHEMBL4595414 0.79 ALDH1A1 (0.43) ALDH1A1KDM4EUSP2HPGDHSD17B10
SCHEMBL4324068 0.78 ALDH1A1 (0.58) CYP2C19ALDH1A1KDM4EUSP2HPGD
SCHEMBL5271103 0.78 AAK1 (0.43) CYP2C19ALDH1A1KDM4EUSP2HPGD
SCHEMBL5176013 0.78 CYP2C19 (0.47) TAS2R14CYP2C19ALDH1A1KDM4EUSP2
SCHEMBL2379685 0.77 ALDH1A1 (0.56) ALDH1A1KDM4EUSP2ESRRAAR
SCHEMBL29546917 0.76 AR (0.52) PTPN1PTPN6PTPN11TAS2R14AR
SCHEMBL12151755 0.76 AR (0.52) PTPN1PTPN6PTPN11TAS2R14AR
SCHEMBL4594851 0.74 PTGDR2 (0.65) PTPN1PTPN6PTPN11TAS2R14PTGDR2
SCHEMBL12818198 0.74 AR (0.45) PTPN1PTPN6PTPN11TAS2R14MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945646-A1 PYRIMIDINE COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS Cellzome (UK) Ltd. (GB) 2008-07-23 EP disclosed
WO-2007039467-A1 PYRIMIDINE COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS CELLZOME (UK) LTD. (GB) 2007-04-12 WO disclosed