SCHEMBL4596868

SCHEMBL4596868

Fc1cc(-c2ccc(C(F)(F)F)cc2)cc2c1NC(=S)NC2.O=C1CCc2cc(-c3ccc(C(F)(F)F)cc3)ccc2N1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 14/20 0.65
PDE3B Q13370 2/20 0.42
PDE3A Q14432 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP11B1 P15538 2/20 0.42
CYP11B2 P19099 2/20 0.42
CYP2C9 P11712 1/20 0.42
TBXAS1 P24557 1/20 0.42
TDP2 O95551 1/20 0.41
AKT1 P31749 1/20 0.41
PKM P14618 1/20 0.40
PKLR P30613 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4890704 0.87 KIF11 (0.41) KIF11TDP2
SCHEMBL1396616 0.81 KIF11 (1.00) KIF11PDE3BPDE3ACYP1A2CYP11B1
SCHEMBL4893178 0.80 KIF11 (0.63) KIF11CYP1A2CYP11B1CYP11B2TDP2
SCHEMBL4897861 0.80 KIF11 (0.72) KIF11PDE3BPDE3ACYP1A2CYP11B1
SCHEMBL4596526 0.78 KIF11 (0.57) KIF11PDE3BPDE3ACYP1A2CYP11B1
SCHEMBL4888035 0.75 KIF11 (0.86) KIF11PDE3BPDE3ACYP1A2CYP11B1
SCHEMBL4888861 0.75 KIF11 (0.86) KIF11PDE3BPDE3ACYP1A2CYP11B1
SCHEMBL4594955 0.74 KIF11 (0.59) KIF11PDE3BPDE3ACYP1A2CYP11B1
SCHEMBL3310186 0.74 KIF11 (0.70) KIF11PDE3BPDE3ACYP1A2CYP11B1
SCHEMBL1903306 0.72 KIF11 (0.80) KIF11PDE3BPDE3ACYP1A2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874753-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113432-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed