SCHEMBL4595397

SCHEMBL4595397

CC(C)(C)C(NC(=O)O)C(O)c1cccc2c1OCO2

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
POLB P06746 2/20 0.41
PPARG P37231 1/20 0.38
TACR1 P25103 5/20 0.37
KDM4C Q9H3R0 1/20 0.36
DRD2 P14416 4/20 0.35
HTR2A P28223 4/20 0.35
DRD3 P35462 4/20 0.35
MGAM O43451 1/20 0.35
AMY1A P0DUB6 1/20 0.35
GAA P10253 1/20 0.35
SI P14410 1/20 0.35
MGAM2 Q2M2H8 1/20 0.35
FAAH O00519 1/20 0.34
MAOB P27338 2/20 0.34
MAPK1 P28482 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19305417 0.75 ALDH1A1 (0.41) ALDH1A1POLBPPARGTACR1KDM4C
SCHEMBL4381017 0.73 ALDH1A1 (0.46) ALDH1A1GAALMNA
SCHEMBL4473207 0.71 ALDH1A1 (0.46) ALDH1A1POLBPPARGTACR1KDM4C
SCHEMBL11756576 0.70 ALDH1A1 (0.42) ALDH1A1POLBPPARGTACR1DRD2
SCHEMBL4380601 0.70 SLC6A4 (0.47) ALDH1A1POLBHTR2AKDM4ELMNA
SCHEMBL19312191 0.69 ALDH1A1 (0.44) ALDH1A1POLBPPARGTACR1DRD2
SCHEMBL4595541 0.69 POLB (0.38) ALDH1A1POLBGAALMNAHPGD
SCHEMBL17724563 0.69 ALDH1A1 (0.39) ALDH1A1POLBTACR1DRD2HTR2A
SCHEMBL7687089 0.69 ALDH1A1 (0.42) ALDH1A1POLBTACR1KDM4CMGAM
SCHEMBL31688946 0.69 ALDH1A1 (0.43) ALDH1A1POLBPPARGTACR1KDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874768-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113837-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed