SCHEMBL4595402

SCHEMBL4595402

CC1Cc2cc(-c3ccccc3)cc(-c3cccc(Cl)c3)c2O1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.39
HTR1A P08908 1/20 0.38
HTR7 P34969 1/20 0.38
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
TSHR P16473 1/20 0.36
NFKB1 P19838 1/20 0.36
RAB9A P51151 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
SLC6A9 P48067 1/20 0.36
TDP2 O95551 2/20 0.36
ADORA1 P30542 2/20 0.36
PARP1 P09874 3/20 0.35
PGR P06401 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596326 0.88 CNR1 (0.41) GRM2HTR1AMAOAMAOBSMN1; SMN2
SCHEMBL4596906 0.85 HTR1A (0.39) GRM2HTR1AHTR7PTGS1PTGS2
SCHEMBL5583521 0.85 NPC1 (0.37) MAOAMAOBSMN1; SMN2NPC1TSHR
SCHEMBL5595946 0.85 S1PR4 (0.39) PTGS2MAOAMAOBSMN1; SMN2NPC1
SCHEMBL4595401 0.84 NPC1 (0.36) GRM2HTR1AHTR7PTGS1PTGS2
SCHEMBL4596409 0.84 PARP1 (0.39) GRM2HTR1AHTR7MAOAMAOB
SCHEMBL5605603 0.84 HTR1A (0.44) GRM2HTR1AHTR7PTGS1PTGS2
SCHEMBL5583714 0.83 CNR1 (0.39) GRM2HTR1AHTR7PTGS1PTGS2
SCHEMBL6047913 0.82 GPR84 (0.45) GRM2HTR1AHTR7SMN1; SMN2NPC1
SCHEMBL5605602 0.82 HTR1A (0.35) GRM2HTR1AHTR7PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP disclosed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO disclosed