SCHEMBL4595401

SCHEMBL4595401

[CH2]C1Cc2cc(-c3ccccc3)cc(-c3cccc(Cl)c3)c2O1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
TP53 P04637 1/20 0.36
TSHR P16473 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ADORA1 P30542 3/20 0.36
TDP2 O95551 2/20 0.36
HTR1A P08908 1/20 0.36
HTR7 P34969 1/20 0.36
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
PGR P06401 1/20 0.35
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
TDO2 P48775 1/20 0.34
ADORA2A P29274 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596319 0.88 CYP1A2 (0.41) NPC1RAB9ASMN1; SMN2PTGS1PTGS2
SCHEMBL5583519 0.84 CNR2 (0.36) NPC1RAB9ATSHRSMN1; SMN2ADORA1
SCHEMBL4596904 0.84 HTR1A (0.38) TP53HTR1AHTR7PTGS1PTGS2
SCHEMBL4595402 0.84 GRM2 (0.39) NPC1RAB9ATP53TSHRNFKB1
SCHEMBL4596405 0.84 HTR1A (0.36) HTR1AHTR7MAOAMAOBPARP10
SCHEMBL5583710 0.83 CYP2A6 (0.39) NPC1RAB9AADORA1HTR1AHTR7
SCHEMBL4595446 0.82 GAA (0.37) HTR1AHTR7TDO2MEN1GAA
SCHEMBL5605603 0.81 HTR1A (0.44) NPC1RAB9ATP53TSHRNFKB1
SCHEMBL4230249 0.81 AQP1 (0.50) NPC1RAB9ATP53TSHRNFKB1
SCHEMBL6047912 0.81 GPR84 (0.41) NPC1RAB9ATP53NFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP disclosed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO disclosed