SCHEMBL4596108

SCHEMBL4596108

Cc1cc2c(c(-c3ccc(Cl)cc3Cl)c1)OC(CCc1ccccc1)C2

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 3/20 0.51
SIRT2 Q8IXJ6 2/20 0.47
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
NPC1 O15118 1/20 0.39
CYP2C19 P33261 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CYP3A4 P08684 2/20 0.37
CXCR2 P25025 1/20 0.36
DRD4 P21917 2/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
CRHR1 P34998 1/20 0.35
EZH2 Q15910 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596987 0.90 SIRT2 (0.55) AQP1SIRT2CYP1A2CYP2D6CYP2C9
SCHEMBL4596777 0.85 SIRT2 (0.49) AQP1SIRT2CYP1A2CYP2D6CYP2C9
SCHEMBL4595484 0.84 AQP1 (0.51) AQP1SIRT2CYP3A4DRD4EZH2
SCHEMBL4225193 0.84 AQP1 (0.61) AQP1SIRT2ALDH1A1EZH2
SCHEMBL4224721 0.82 AQP1 (0.74) AQP1CRHR1EZH2
SCHEMBL6367685 0.81 AQP1 (0.46) AQP1
SCHEMBL4225189 0.80 AQP1 (0.77) AQP1CYP1A2NPC1CYP2C19RAB9A
SCHEMBL4596103 0.80 AQP1 (0.43) AQP1CYP1A2CYP2D6CYP2C9NPC1
SCHEMBL4225381 0.78 AQP1 (0.59) AQP1CYP1A2NPC1CYP2C19RAB9A
SCHEMBL4790525 0.78 AQP1 (0.56) AQP1SIRT2NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed