SCHEMBL4595484

SCHEMBL4595484

Cc1cc2c(c(-c3c(Cl)cccc3Cl)c1)OC(CCc1ccccc1)C2

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 3/20 0.51
SIRT2 Q8IXJ6 3/20 0.48
CYP3A4 P08684 1/20 0.39
EZH2 Q15910 1/20 0.34
SSTR2 P30874 1/20 0.34
SSTR4 P31391 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
DRD4 P21917 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4225698 0.85 AQP1 (0.54) AQP1SIRT2EZH2SSTR2SSTR4
SCHEMBL4596679 0.84 SIRT2 (0.50) AQP1SIRT2CYP3A4SSTR2SSTR4
SCHEMBL4596108 0.84 AQP1 (0.51) AQP1SIRT2CYP3A4EZH2DRD4
SCHEMBL4596497 0.84 SIRT2 (0.56) AQP1SIRT2CYP3A4EZH2SSTR2
SCHEMBL4220310 0.82 AQP1 (0.56) AQP1SIRT2EZH2SSTR2SSTR4
SCHEMBL4596351 0.80 AQP1 (0.45) AQP1
SCHEMBL4595085 0.80 SIRT2 (0.54) AQP1SIRT2CYP3A4EZH2SSTR2
SCHEMBL4225690 0.80 AQP1 (0.77) AQP1SIRT2CYP3A4EZH2SLC6A2
SCHEMBL4232694 0.79 AQP1 (0.58) AQP1SIRT2CYP3A4EZH2
SCHEMBL4595481 0.79 AQP1 (0.43) AQP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed