SCHEMBL4596375

SCHEMBL4596375

O=C1NCc2cc(-c3ccc(C(F)(F)F)cc3)ccc2N1Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 1/20 0.47
GSK3B P49841 1/20 0.47
CHRM5 P08912 4/20 0.43
NPSR1 Q6W5P4 1/20 0.43
KIF11 P52732 2/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
POLB P06746 1/20 0.41
MDH2 P40926 1/20 0.41
TDP2 O95551 1/20 0.41
CHRM4 P08173 1/20 0.41
SIGMAR1 Q99720 1/20 0.40
CFTR P13569 1/20 0.40
HSP90AA1 P07900 1/20 0.40
CXCR2 P25025 1/20 0.40
TACR1 P25103 1/20 0.39
HIF1A Q16665 1/20 0.38
EPAS1 Q99814 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4896274 0.86 CHRM5 (0.43) GSK3AGSK3BCHRM5HSP90AA1
SCHEMBL1862096 0.77 GSK3A (0.56) GSK3AGSK3BPOLBMDH2
SCHEMBL30806297 0.76 GSK3A (0.55) GSK3AGSK3BPOLB
SCHEMBL29558351 0.75 GSK3A (0.65) GSK3AGSK3BCHRM5DRD2DRD4
SCHEMBL4791747 0.75 GSK3A (0.65) GSK3AGSK3BCHRM5DRD2DRD4
SCHEMBL3310868 0.74 HDAC6 (0.53) NPSR1POLB
SCHEMBL27376904 0.72 CASP1 (0.57) GSK3AGSK3B
SCHEMBL30806305 0.72 CASP1 (0.57) GSK3AGSK3B
SCHEMBL13330272 0.72 HSP90AA1 (0.53) CHRM5NPSR1POLBHSP90AA1
SCHEMBL3304528 0.72 PRKAG1 (0.49) POLBTACR1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080176830-A1 Compounds, Compositions, and Methods ADAMS NICHOLAS D 2008-07-24 US claimed
US-20080176830-A1 Compounds, Compositions, and Methods ADAMS NICHOLAS D 2008-07-24 US disclosed
US-20080176830-A1 Compounds, Compositions, and Methods ADAMS NICHOLAS D 2008-07-24 US disclosed
EP-1874753-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113432-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080176830-A1 Compounds, Compositions, and Methods ALPP, PCNA, MKI67 GSK3A 1510/4885GSK3B 1444/4885CHRM5 4270/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.