SCHEMBL4596542

SCHEMBL4596542

COc1ccccc1C(OCc1ccccc1)C(C)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
ACHE P22303 1/20 0.45
HTT P42858 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
POLB P06746 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
HTR1A P08908 2/20 0.43
ADRA1D P25100 2/20 0.43
ADRA1A P35348 2/20 0.43
ADRA1B P35368 2/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
TDP1 Q9NUW8 2/20 0.42
RCE1 Q9Y256 1/20 0.42
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
SGMS2 Q8NHU3 1/20 0.41
RXRA P19793 1/20 0.40
CASR P41180 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596807 0.88 SMN1; SMN2 (0.41) CA1CA2ACHEHTTL3MBTL1
SCHEMBL5186083 0.86 GAA (0.40) CA1CA2ACHEPOLBRCE1
SCHEMBL5186091 0.85 MEN1 (0.43) CA1CA2ACHEHTTL3MBTL1
SCHEMBL5653055 0.83 CA1 (0.46) CA1CA2ACHEHTTL3MBTL1
SCHEMBL4944038 0.79 CA1 (0.43) CA1CA2ACHEHTTL3MBTL1
SCHEMBL27586977 0.76 KMT2A (0.42) CA1CA2ACHEHTTPOLB
SCHEMBL28769510 0.74 SGMS2 (0.56) L3MBTL1HTR1AADRA1DADRA1AADRA1B
SCHEMBL21980698 0.74 ATM (0.48) CA1CA2L3MBTL1TDP1KDM4E
SCHEMBL17901117 0.74 ATM (0.48) CA1CA2L3MBTL1TDP1KDM4E
SCHEMBL19714109 0.74 ATM (0.48) CA1CA2L3MBTL1TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed
EP-1802598-A2 ASYMMETRIC SYNTHESIS OF DIHYDROBENZOFURAN DERIVATIVES Wyeth a Corporation of the State of Delaware (US) 2007-07-04 EP disclosed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP disclosed
WO-2006047288-A2 ASYMMETRIC SYNTHESIS OF DIHYDROBENZOFURAN DERIVATIVES WYETH (US) 2006-05-04 WO disclosed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO disclosed