SCHEMBL4596807

SCHEMBL4596807

COc1ccc(F)cc1C(OCc1ccccc1)C(C)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.41
NR3C1 P04150 2/20 0.40
FFAR1 O14842 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
ACHE P22303 2/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
MGAM O43451 1/20 0.39
GAA P10253 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
NPC1 O15118 1/20 0.39
HPGD P15428 1/20 0.39
RAB9A P51151 1/20 0.39
PSMB5 P28074 1/20 0.39
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596542 0.88 CA1 (0.45) CA1CA2ACHECYP2C19POLB
SCHEMBL5186083 0.86 GAA (0.40) SMN1; SMN2CA1CA2ACHEMGAM
SCHEMBL5186091 0.85 MEN1 (0.43) SMN1; SMN2CA1CA2ACHEMGAM
SCHEMBL5653055 0.76 CA1 (0.46) CA1CA2ACHECYP2C19GAA
SCHEMBL6255859 0.75 CYP2C19 (0.49) SMN1; SMN2NR3C1FFAR1FFAR4CYP3A4
SCHEMBL5186024 0.74 HTR1A (0.33) SMN1; SMN2MGAMGAASIMGAM2
SCHEMBL18908296 0.73 ALDH1A1 (0.39) SMN1; SMN2NR3C1FFAR1FFAR4CA1
SCHEMBL18908273 0.73 ALDH1A1 (0.39) SMN1; SMN2NR3C1FFAR1FFAR4CA1
SCHEMBL2588953 0.72 ADRA2A (0.45) HTR2AHTR2CADRA1A
SCHEMBL2592419 0.72 ADRA2A (0.45) HTR2AHTR2CADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed
EP-1802598-A2 ASYMMETRIC SYNTHESIS OF DIHYDROBENZOFURAN DERIVATIVES Wyeth a Corporation of the State of Delaware (US) 2007-07-04 EP disclosed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP disclosed
WO-2006047288-A2 ASYMMETRIC SYNTHESIS OF DIHYDROBENZOFURAN DERIVATIVES WYETH (US) 2006-05-04 WO disclosed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO disclosed