SCHEMBL4596827

SCHEMBL4596827

Cc1ccc(Cl)cc1-c1cc(F)cc2c1O[C@H](C)C2

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 3/20 0.53
PARP1 P09874 4/20 0.45
L3MBTL1 Q9Y468 1/20 0.39
BRD4 O60885 2/20 0.34
AGPAT2 O15120 1/20 0.32
HTR1A P08908 1/20 0.32
IDO1 P14902 1/20 0.31
CREBBP Q92793 1/20 0.31
AR P10275 3/20 0.31
PDE2A O00408 1/20 0.31
PDE10A Q9Y233 1/20 0.31
CETP P11597 1/20 0.31
SLC6A4 P31645 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4764345 0.90 AQP1 (0.56) AQP1PARP1L3MBTL1BRD4HTR1A
SCHEMBL4713102 0.88 AQP1 (0.54) AQP1PARP1L3MBTL1BRD4HTR1A
SCHEMBL4596815 0.86 PARP1 (0.47) AQP1PARP1BRD4CREBBP
SCHEMBL4596825 0.86 AQP1 (0.52) AQP1PARP1L3MBTL1AGPAT2IDO1
SCHEMBL4712234 0.85 AQP1 (0.67) AQP1PARP1BRD4HTR1ACREBBP
SCHEMBL4230928 0.84 AQP1 (0.76) AQP1PARP1L3MBTL1AGPAT2SLC6A4
SCHEMBL5605564 0.84 AQP1 (0.56) AQP1L3MBTL1AGPAT2IDO1
SCHEMBL14113171 0.84 AQP1 (0.76) AQP1PARP1L3MBTL1AGPAT2SLC6A4
SCHEMBL4230233 0.84 AQP1 (0.59) AQP1L3MBTL1AGPAT2PDE2APDE10A
SCHEMBL4606791 0.84 AQP1 (0.47) AQP1PARP1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed