SCHEMBL4596938

SCHEMBL4596938

Fc1cccc(F)c1-c1cccc2c1OCC2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.45
GRM2 Q14416 1/20 0.37
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
RORC P51449 1/20 0.34
SRD5A1 P18405 1/20 0.33
HTR1A P08908 1/20 0.33
HASPIN Q8TF76 1/20 0.33
CYP19A1 P11511 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
MAP4K1 Q92918 1/20 0.32
PDE4B Q07343 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
KCNH2 Q12809 1/20 0.32
HTR7 P34969 1/20 0.32
NOTUM Q6P988 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29791283 0.83 PARP1 (0.52) PARP1RORCHTR1ACYP19A1SLC6A2
SCHEMBL13635655 0.83 PARP1 (0.52) PARP1RORCHTR1ACYP19A1SLC6A2
SCHEMBL8248843 0.80 LMNA (0.36) PARP1HTR1A
SCHEMBL1840365 0.77 PARP1 (0.44) PARP1GRM2GSK3AGSK3BHASPIN
SCHEMBL8255618 0.77 HTR7 (0.46) HTR1AHTR7
SCHEMBL28230835 0.74 PARP1 (0.47) PARP1GRM2HTR1ASLC6A2SLC6A4
SCHEMBL1812982 0.72 ACHE (0.42) PARP1HTR1A
SCHEMBL20713018 0.71 PARP1 (0.45) PARP1GRM2HASPINSLC6A2SLC6A4
SCHEMBL27896035 0.71 KCNH2 (0.43) PARP1SLC6A2SLC6A4KCNH2
SCHEMBL14786485 0.70 CDK2 (0.44) PARP1GRM2RORCHASPINMAP4K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed