SCHEMBL4596940

SCHEMBL4596940

Cc1cccc([C@@H]2CNC(=O)N2C2CCN(C(=O)O)CC2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
ADAM17 P78536 1/20 0.38
ADAMTS5 Q9UNA0 1/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD11B1 P28845 2/20 0.37
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
DRD3 P35462 1/20 0.37
FAAH O00519 1/20 0.37
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
CHRM1 P11229 1/20 0.37
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5576017 0.85 GPR119 (0.53) HDAC1HDAC6KMT2ATP53MAPT
SCHEMBL5576012 0.85 GPR119 (0.53) HDAC1HDAC6KMT2ATP53MAPT
SCHEMBL4597772 0.82 HTR2C (0.52) HDAC1HDAC6KMT2ATP53MAPT
SCHEMBL4597778 0.82 HTR2C (0.52) HDAC1HDAC6KMT2ATP53MAPT
SCHEMBL4552094 0.76 CCR5 (0.49) CCR5
SCHEMBL4597324 0.74 GPR119 (0.51) KMT2ATP53MAPTMEN1KDM4E
SCHEMBL4610243 0.67 SLC18A3 (0.44) KMT2ASMN1; SMN2MEN1
SCHEMBL3815926 0.67 SLC18A3 (0.44) KMT2ASMN1; SMN2MEN1
SCHEMBL27341297 0.67 PRMT5 (0.49) ADAM17HSD11B1
SCHEMBL4597612 0.67 GPR119 (0.52) HDAC1HDAC6KMT2ATP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed