SCHEMBL4596993

SCHEMBL4596993

O=c1[nH]c(C2CN(c3ccc(CN4CCOCC4)cc3)C2)cc2c1cnn2-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.44
ALDH1A1 P00352 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPK1 P28482 2/20 0.40
TNKS O95271 1/20 0.40
CCR5 P51681 1/20 0.40
BTK Q06187 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CDK4 P11802 1/20 0.39
CCND1 P24385 1/20 0.39
CDK2 P24941 1/20 0.39
ENPP2 Q13822 4/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
PDE9A O76083 2/20 0.38
PDE1C Q14123 1/20 0.38
KDM4E B2RXH2 1/20 0.38
USP2 O75604 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4502011 0.82 MAPK1 (0.50) PARP1ALDH1A1MAPK1LMNAMAPT
SCHEMBL4514708 0.70 MAPK1 (0.49) ALDH1A1MAPK1LMNAMAPTPDE9A
SCHEMBL4502316 0.70 PDE9A (0.47) TNKSPDE9APDE1C
SCHEMBL4502003 0.69 PDE9A (0.57) PDE9APDE1C
SCHEMBL22042885 0.67 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL4504690 0.66 TYK2 (0.49) ALDH1A1SMN1; SMN2MAPK1NPC1LMNA
SCHEMBL4591180 0.65 TYK2 (0.62) ALDH1A1SMN1; SMN2MAPK1NPC1RAB9A
SCHEMBL16728898 0.64 RAB9A (0.52) ALDH1A1RAB9AMAPTKDM4ETSHR
SCHEMBL4516124 0.64 TYK2 (0.54) ALDH1A1MAPK1MAPTPDE9APDE1C
SCHEMBL27704094 0.62 MAPK10 (0.41) ALDH1A1LMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008055959-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2008-05-15 WO disclosed