SCHEMBL4597250

SCHEMBL4597250

Cc1ccc(-c2cc(F)c3c(c2)CC(C)O3)cc1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.40
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
BRD4 O60885 2/20 0.34
KDM4E B2RXH2 1/20 0.33
CREBBP Q92793 1/20 0.33
HTR1A P08908 4/20 0.32
FFAR4 Q5NUL3 2/20 0.32
TDP1 Q9NUW8 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596976 0.89 PARP1 (0.44) PARP1NPC1RAB9ABRD4HTR1A
SCHEMBL5583554 0.87 PARP1 (0.40) PARP1NPC1RAB9ABRD4HTR1A
SCHEMBL4597169 0.84 KDM4E (0.40) PARP1NPC1RAB9ABRD4KDM4E
SCHEMBL4595479 0.84 PARP1 (0.38) PARP1MAOAMAOBNPC1RAB9A
SCHEMBL4597245 0.84 FFAR4 (0.31) FFAR4PDE3BPDE3A
SCHEMBL4222492 0.80 PRKAB2 (0.51) MAOB
SCHEMBL4595107 0.79 PARP1 (0.42) PARP1HTR1A
SCHEMBL5583539 0.78 HPRT1 (0.47) PARP1MAOAMAOBNPC1RAB9A
SCHEMBL4596609 0.78 PARP1 (0.38) PARP1MAOAMAOBNPC1RAB9A
SCHEMBL4596742 0.78 PARP1 (0.49) PARP1MAOAMAOBBRD4HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007509174-A 2007-04-12 JP claimed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP claimed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO claimed
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed