SCHEMBL5583554

SCHEMBL5583554

CC1Cc2cc(-c3ccc(Cl)cc3)cc(F)c2O1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.40
GRM2 Q14416 2/20 0.36
HTR2A P28223 2/20 0.36
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
HTR1A P08908 2/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
AHR P35869 1/20 0.33
AQP1 P29972 2/20 0.33
BRD4 O60885 1/20 0.32
CHRM1 P11229 1/20 0.31
MCHR1 Q99705 1/20 0.31
PTGS2 P35354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596976 0.88 PARP1 (0.44) PARP1GRM2HTR2ANPC1RAB9A
SCHEMBL4597250 0.87 PARP1 (0.40) PARP1NPC1RAB9AHTR1ABRD4
SCHEMBL4597572 0.85 GRM2 (0.40) PARP1GRM2HTR1A
SCHEMBL4597169 0.83 KDM4E (0.40) PARP1GRM2NPC1RAB9ABRD4
SCHEMBL5583552 0.82 AHR (0.33) AHRAQP1
SCHEMBL4706710 0.79 CNR1 (0.39) PARP1GRM2NPC1RAB9AHTR1A
SCHEMBL4596326 0.79 CNR1 (0.41) PARP1GRM2NPC1RAB9AHTR1A
SCHEMBL4230632 0.79 AQP1 (0.54) PARP1GRM2HTR2AAHRAQP1
SCHEMBL4963750 0.78 PARP1 (0.48) PARP1GRM2HTR2AHTR1ACNR1
SCHEMBL4595107 0.78 PARP1 (0.42) PARP1GRM2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007509174-A 2007-04-12 JP claimed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP claimed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO claimed