SCHEMBL4597245

SCHEMBL4597245

[CH2]C1Cc2cc(-c3ccc(C)cc3)cc(F)c2O1

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 1/20 0.31
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596968 0.88 KDM1A (0.36)
SCHEMBL5583552 0.85 AHR (0.33)
SCHEMBL4597165 0.85 NPC1 (0.37)
SCHEMBL4595474 0.85 PARP10 (0.34) PDE3BPDE3A
SCHEMBL4597250 0.84 PARP1 (0.40) FFAR4PDE3BPDE3A
SCHEMBL4596607 0.79 PRKAB2 (0.35) PDE3BPDE3A
SCHEMBL4222492 0.79 PRKAB2 (0.51)
SCHEMBL5583536 0.79 HPRT1 (0.46)
SCHEMBL4596739 0.78 AQP1 (0.38)
SCHEMBL4595105 0.78 TAAR1 (0.36) PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007509174-A 2007-04-12 JP claimed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP claimed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO claimed
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed