SCHEMBL4598133

SCHEMBL4598133

O=C1CN(OC(=O)C(F)(F)F)C(=O)N1CCOc1ccc(-c2ccccc2F)nc1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PLA2G7 Q13093 1/20 0.39
RAB9A P51151 2/20 0.37
NPC1 O15118 1/20 0.37
PDK2 Q15119 1/20 0.35
IL4I1 Q96RQ9 1/20 0.34
WNT3A P56704 11/20 0.33
HPGD P15428 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
DHODH Q02127 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4598130 0.79 NPC1 (0.38) RAB9ANPC1PDK2WNT3A
SCHEMBL4590822 0.79 RAB9A (0.47) PLA2G7RAB9ANPC1PDK2IL4I1
SCHEMBL4590531 0.76 RAB9A (0.63) RAB9ANPC1HPGDNPSR1
SCHEMBL4590799 0.76 RAB9A (0.44) PLA2G7RAB9ANPC1IL4I1HPGD
SCHEMBL4590767 0.73 PDK2 (0.47) PLA2G7RAB9ANPC1PDK2
SCHEMBL3182212 0.71 NPC1 (0.39) RAB9ANPC1PDK2WNT3AHPGD
SCHEMBL4590673 0.70 PDK2 (0.52) RAB9ANPC1PDK2IL4I1
SCHEMBL4590073 0.70 MTNR1A (0.55) RAB9ANPC1PDK2HPGD
SCHEMBL4590077 0.70 RAB9A (0.41) RAB9ANPC1PDK2HPGDNPSR1
SCHEMBL12020957 0.69 NPC1 (0.52) RAB9ANPC1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899321-A1 HETEROARYL-SUBSTITUTED AMIDES COMPRISING A SATURATED LINKER GROUP, AND THEIR USE AS PHARMACEUTICALS Sanofi-Aventis (FR) 2008-03-19 EP disclosed
WO-2007000246-A1 HETEROARYL-SUBSTITUTED AMIDES COMPRISING A SATURATED LINKER GROUP, AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS (DE) 2007-01-04 WO disclosed