SCHEMBL4601231

SCHEMBL4601231

Cc1ccccc1-c1ccc(C(=O)NCc2cccc(Cl)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.55
NPC1 O15118 1/20 0.53
DRD2 P14416 1/20 0.53
CNR2 P34972 2/20 0.52
MAPK14 Q16539 1/20 0.52
CXCR3 P49682 1/20 0.52
EGFR P00533 1/20 0.51
PLA2G1B P04054 1/20 0.51
HTT P42858 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
ATG4B Q9Y4P1 1/20 0.51
MEN1 O00255 1/20 0.51
HCRTR1 O43613 1/20 0.51
KMT2A Q03164 1/20 0.51
CNR1 P21554 3/20 0.51
ROCK2 O75116 1/20 0.51
ROCK1 Q13464 1/20 0.51
MAPK1 P28482 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4601230 0.87 ROCK2 (0.57) PPARGNPC1DRD2CNR2EGFR
SCHEMBL2912888 0.86 MAPK1 (0.55) PPARGNPC1MAPK14CXCR3CNR1
SCHEMBL30462959 0.83 NPC1 (0.61) NPC1MAPK14CXCR3HTTMEN1
SCHEMBL13947495 0.83 NPC1 (0.61) NPC1MAPK14CXCR3HTTMEN1
SCHEMBL3461102 0.81 NPC1 (0.70) PPARGNPC1CXCR3HTTMEN1
SCHEMBL24628975 0.81 ROCK2 (0.62) NPC1CXCR3EGFRROCK2ROCK1
SCHEMBL3028316 0.81 HDAC1 (0.71) NPC1CXCR3EGFRROCK2ROCK1
SCHEMBL4859805 0.80 MAPK14 (0.80) MAPK14
SCHEMBL6605534 0.80 MAPK14 (0.80) MAPK14
SCHEMBL2345084 0.79 MAPK14 (0.66) MAPK14MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940786-A1 BIPHENYL DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C Arrow Therapeutics Limited (GB) 2008-07-09 EP disclosed
WO-2007031791-A1 BIPHENYL DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C ARROW THERAPEUTICS LIMITED (GB) 2007-03-22 WO disclosed