SCHEMBL4602335

SCHEMBL4602335

C=C(C(=O)O)c1ccc(OCCOC)cc1Oc1ncc(Br)cc1C

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.38
TDP1 Q9NUW8 1/20 0.38
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.36
AAK1 Q2M2I8 1/20 0.36
PPARG P37231 7/20 0.34
CHEK2 O96017 1/20 0.33
HPGD P15428 1/20 0.33
LSS P48449 2/20 0.33
CNR2 P34972 1/20 0.33
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4602334 0.81 EGFR (0.37) KDM4ELMNACYP1A2CYP3A4CYP2C9
SCHEMBL3205613 0.79 PPARG (0.47) KDM4ELMNACYP1A2CYP3A4CYP2C9
SCHEMBL3205624 0.79 PPARG (0.47) KDM4ELMNACYP1A2CYP3A4CYP2C9
SCHEMBL4602178 0.71 EGFR (0.43) KDM4ELMNAKMT2AAAK1ALDH1A1
SCHEMBL1816280 0.70 TSHR (0.40) KDM4ELMNACYP1A2CYP3A4CYP2C9
SCHEMBL27009298 0.68 ALDH1A1 (0.54) KDM4ELMNAKMT2AALDH1A1
SCHEMBL1505065 0.67 CNR2 (0.48) KMT2AHPGDCNR2ALDH1A1
SCHEMBL16510360 0.67 KDM4E (0.49) KDM4ETDP1HTTHPGD
SCHEMBL3199078 0.67 PPARG (0.49) KDM4EKMT2APPARGCHEK2ALDH1A1
SCHEMBL3199101 0.67 PPARG (0.49) KDM4EKMT2APPARGCHEK2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912645-A2 THERAPEUTIC AGENT FOR DIABETES Takeda Pharmaceutical Company Limited (JP) 2008-04-23 EP disclosed
WO-2007018314-A2 THERAPEUTIC AGENT FOR DIABETES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-15 WO disclosed