SCHEMBL4602334

SCHEMBL4602334

C=CC(=O)Oc1ccc(OCCOC)cc1Oc1ncc(Br)cc1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.37
LMNA P02545 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HTT P42858 1/20 0.37
BTK Q06187 4/20 0.35
PPARG P37231 3/20 0.34
ITK Q08881 2/20 0.34
JAK2 O60674 1/20 0.34
LYN P07948 1/20 0.34
TEC P42680 1/20 0.34
TXK P42681 1/20 0.34
BMX P51813 1/20 0.34
JAK3 P52333 1/20 0.34
CD69 Q07108 1/20 0.34
KDM4E B2RXH2 3/20 0.34
KMT2A Q03164 1/20 0.34
AAK1 Q2M2I8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4602178 0.82 EGFR (0.43) EGFRLMNABTKITKJAK2
SCHEMBL4602335 0.81 KDM4E (0.38) LMNACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL3205613 0.78 PPARG (0.47) LMNACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL3205624 0.78 PPARG (0.47) LMNACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4631636 0.72 PDE4B (0.43) EGFR
SCHEMBL12796997 0.71 THRB (0.54) EGFR
SCHEMBL4632439 0.71 PDE4D (0.42)
SCHEMBL4602781 0.70 EGFR (0.45) EGFRBTKITKJAK2LYN
SCHEMBL1816280 0.69 TSHR (0.40) LMNACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL19564418 0.68 THRB (0.46) EGFRCYP3A4BTKITKJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912645-A2 THERAPEUTIC AGENT FOR DIABETES Takeda Pharmaceutical Company Limited (JP) 2008-04-23 EP disclosed
WO-2007018314-A2 THERAPEUTIC AGENT FOR DIABETES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-15 WO disclosed